Concepedia

Discovery of a small molecule RXFP3/4 agonist that increases food intake in rats upon acute central administration

Brian A. DeChristopher, Soo-Hee Park, Linh Vong, D G Bamford, Hyun-Hee Cho, Rohit Duvadie, Allison Fedolak, Christopher M. Hogan, Toshiyuki Honda, Pramod S. Pandey,

Bioorganic & Medicinal Chemistry Letters · 2019 · 28 citations · 10 references

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10

Insulin-like peptide 5 is an orexigenic gastrointestinal hormone

Johannes Grosse, Helen Heffron, Keith Burling et al. · Proceedings of the National Academy of Sciences · 2014 · 146 citations · Full text

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Relaxin-3:  Improved Synthesis Strategy and Demonstration of Its High-Affinity Interaction with the Relaxin Receptor LGR7 Both<i>In Vitro</i>and<i>In Vivo</i>

Ross A. D. Bathgate, Feng Lin, Nicola F. Hanson et al. · Biochemistry · 2005 · 145 citations

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Synthesis, Conformation, and Activity of Human Insulin‐Like Peptide 5 (INSL5)

Mohammed Akhter Hossain, Ross A. D. Bathgate, Fazel Shabanpoor et al. · ChemBioChem · 2008 · 85 citations · Full text

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The insulinotrophic effect of insulin-like peptide 5 <i>in vitro</i> and <i>in vivo</i>

Xiao Luo, Ting Li, Yue Zhu et al. · Biochemical Journal · 2014 · 53 citations

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Structure of the R3/I5 Chimeric Relaxin Peptide, a Selective GPCR135 and GPCR142 Agonist

Linda M. Haugaard‐Kedström, Mohammed Akhter Hossain, Norelle L. Daly et al. · Journal of Biological Chemistry · 2008 · 47 citations · Full text

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