Concepedia

Synthesis and biological evaluation of some N-(3-(1H-tetrazol-5-yl) phenyl)acetamide derivatives as novel non-carboxylic PTP1B inhibitors designed through bioisosteric modulation

Neelesh Maheshwari, Chandrabose Karthikeyan, Shraddha V. Bhadada, Chandan Sahi, Amit K. Verma, N. S. Hari Narayana Moorthy, Piyush Trivedi

Bioorganic Chemistry · 2018 · 18 citations · 14 references

DOI

Concepts

References

14

Glide:  A New Approach for Rapid, Accurate Docking and Scoring. 1. Method and Assessment of Docking Accuracy

Richard A. Friesner, Jay L. Banks, Robert B. Murphy et al. · Journal of Medicinal Chemistry · 2004 · 9.9K citations

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Global Burden of Diabetes, 1995–2025: Prevalence, numerical estimates, and projections

Hilary King, Ronald E. Aubert, William H. Herman · Diabetes Care · 1998 · 6.3K citations

, , +14

Obesity

David W. Haslam, W. P. T. James · The Lancet · 2005 · 3.8K citations

, , +8

Increased Energy Expenditure, Decreased Adiposity, and Tissue-Specific Insulin Sensitivity in Protein-Tyrosine Phosphatase 1B-Deficient Mice

Lori D. Klaman, Olivier Boss, Odile D. Peroni et al. · Molecular and Cellular Biology · 2000 · 1.2K citations

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Molecular Basis for the Dephosphorylation of the Activation Segment of the Insulin Receptor by Protein Tyrosine Phosphatase 1B

Annette Salmeen, Jannik N. Andersen, Michael P. Myers et al. · Molecular Cell · 2000 · 464 citations · Full text

, , +17