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Bioisosteres of ethyl 8-ethynyl-6-(pyridin-2-yl)-4H-benzo[f]imidazo [1,5-a][1,4]diazepine-3-carboxylate (HZ-166) as novel alpha 2,3 selective potentiators of GABAA receptors: Improved bioavailability enhances anticonvulsant efficacy

Selective PotentiatorsFunctional SelectivityMedicineBioavailability EnhancesMechanism Of ActionPharmacological AgentNeuropharmacologyPharmacotherapyNeurosciencePharmacologyGabaa ReceptorsDrug Discovery