Concepedia

Design, synthesis and biological evaluation of novel 7-azaspiro[3.5]nonane derivatives as GPR119 agonists

Daisuke Matsuda, Madoka Kawamura, Yohei Kobashi, Fumiyasu Shiozawa, Youichirou Suga, Keiko Fusegi, Shinichi Nishimoto, Kayo Kimura, Masako Miyoshi, Noriko Takayama,

Bioorganic & Medicinal Chemistry · 2018 · 12 citations · 16 references

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16

Escape from Flatland: Increasing Saturation as an Approach to Improving Clinical Success

Frank Lovering, Jack Bikker, Christine Humblet · Journal of Medicinal Chemistry · 2009 · 4.4K citations

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Evaluation of Various Dissolution Media for Predicting In Vivo Performance of Class I and II Drugs

Eric Galia, Eleftheria Nicolaides, D. Hörter et al. · Pharmaceutical Research · 1998 · 923 citations

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Glucagon-Like Peptide 1 Inhibits Cell Apoptosis and Improves Glucose Responsiveness of Freshly Isolated Human Islets

Loredana Farilla, Angela Bulotta, Boaz Hirshberg et al. · Endocrinology · 2003 · 668 citations

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Glycemic Control From 1988 to 2000 Among U.S. Adults Diagnosed With Type 2 Diabetes

Carol E. Koro, Steven J. Bowlin, Nancy Bourgeois et al. · Diabetes Care · 2004 · 654 citations · Full text

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Deorphanization of a G protein-coupled receptor for oleoylethanolamide and its use in the discovery of small-molecule hypophagic agents

Hilary A. Overton, Adam J. Babbs, S. M. Doel et al. · Cell Metabolism · 2006 · 648 citations · Full text

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