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Aryl thiosemicarbazones for the treatment of trypanosomatidic infections

Pasquale Linciano, Carolina Borsoi Moraes, Laura Maria Alcântara, Caio Haddad Franco, Bruno S. Pascoalino, Lúcio H. Freitas-Júnior, Sara Macedo, Nuno Santarém, Anabela Cordeiro‐da‐Silva, Sheraz Gul,

European Journal of Medicinal Chemistry · 2018 · 41 citations · 25 references

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References

25

Human African trypanosomiasis

Reto Brun, Johannes Blum, François Chappuis et al. · The Lancet · 2009 · 915 citations

Synthesis and Structure−Activity Relationship Study of Potent Trypanocidal Thio Semicarbazone Inhibitors of the Trypanosomal Cysteine Protease Cruzain

Xiaohui Du, Chun Guo, Elizabeth Hansell et al. · Journal of Medicinal Chemistry · 2002 · 383 citations · Full text

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Synthesis and Structure−Activity Relationships of Parasiticidal Thiosemicarbazone Cysteine Protease Inhibitors against <i>Plasmodium falciparum</i>, <i>Trypanosoma brucei</i>, and <i>Trypanosoma cruzi</i>

Doron C. Greenbaum, Zachary B. Mackey, Elizabeth Hansell et al. · Journal of Medicinal Chemistry · 2004 · 254 citations · Full text

, , +17

Nitroheterocyclic compounds are more efficacious than CYP51 inhibitors against Trypanosoma cruzi: implications for Chagas disease drug discovery and development

Carolina Borsoi Moraes, Miriam A. Giardini, Hwayoung Kim et al. · Scientific Reports · 2014 · 208 citations · Full text

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PTR1: a reductase mediating salvage of oxidized pteridines and methotrexate resistance in the protozoan parasite Leishmania major.

Alexandre Ribeiro Bello, Bakela Nare, D. Freedman et al. · Proceedings of the National Academy of Sciences · 1994 · 192 citations

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