Concepedia

Cu/Pd cooperatively catalyzed tandem intramolecular anti-Markovnikov hydroarylation of unsaturated amides: facile construction of 3,4-dihydroquinolinones <i>via</i> borylation/intramolecular C(sp<sup>3</sup>)–C(sp<sup>2</sup>) cross coupling

Zhijie Kuang, Bingnan Li, Qiuling Song

Chemical Communications · 2017 · 41 citations · 33 references

DOI

Concepts

Abstract

cross-coupling has been disclosed. 3,4-Dihydroquinolinones, one type of important scaffold prevailing in pharmaceuticals and biologically active compounds, could be readily accessible with high regio-selectivity and high yields.

References

33

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