Bioorganic & Medicinal Chemistry · 2017 · 27 citations · 26 references
PharmacyMedicinal ChemistryPharmacologyDrug DiscoveryProdrug DesignRheumatologyPeptide ProdrugsPh-activated ProdrugsProdrug Activation MechanismsRheumatoid ArthritisEnzymatic InhibitionPh-dependent ActivationPh-dependent RegulationPka-driven Prodrug DesignProdrug Design For SolubilityProdrug Stability AssessmentProdrug Stability Optimization
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Substituted benzimidazoles inhibit gastric acid secretion by blocking (H+ + K+) ATPase
E. Fellenius, T. Berglindh, George Sachs et al. · Nature · 1981 · 625 citations
Medicine, Biochemistry, Pharmacology +10
The mechanism of action of the antisecretory agent omeprazole
P. A. P. Lindberg, Peter Nordberg, Tomas Alminger et al. · Journal of Medicinal Chemistry · 1986 · 307 citations
Kamlesh Dhalwal, Vaibhav Shinde, Yogesh S Biradar et al. · Journal of Food Composition and Analysis · 2008 · 138 citations