Bioorganic & Medicinal Chemistry Letters · 2017 · 51 citations · 18 references
PharmacyMedicinal ChemistryPharmacologyDrug DesignDrug DiscoveryStructure-activity RelationshipsEnzyme InhibitionHit-to-lead OptimizationLead Compound DesignLigand-based DesignPotency OptimizationStructure-activity Relationship AnalysisChemical Synthesis Of AnaloguesEnzyme Inhibitor DiscoveryEnzyme Inhibitor SynthesisLipase InhibitionLipase InhibitorsMedicinal Chemistry ApplicationsMolecular Docking Of InhibitorsMolecular Property-based Design
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Structure of human pancreatic lipase
F.K. Winkler, A. D’Arcy, Willi Hunziker · Nature · 1990 · 1.2K citations
Structure of the pancreatic lipase–procolipase complex
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