Concepedia

Part I: Design, synthesis and biological evaluation of novel pyrazole-benzimidazole conjugates as checkpoint kinase 2 (Chk2) inhibitors with studying their activities alone and in combination with genotoxic drugs

Ahmed S. Abdelsamie, Samia A. Shouman, Yasmin M. Attia, Hamed I. Ali, Ashraf A. Tabll, Reem El‐Shenawy, Yasmine S. El, Mamdouh M. Ali, Abeer E. Mahmoud, Abeer H. Abdel-Halim,

European Journal of Medicinal Chemistry · 2017 · 44 citations · 23 references

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References

23

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Improved protein–ligand docking using GOLD

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Efficacy, safety, and survival with ruxolitinib in patients with myelofibrosis: results of a median 3-year follow-up of COMFORT-I

Srđan Verstovšek, Ruben A. Mesa, Jason Gotlib et al. · Haematologica · 2015 · 329 citations · Full text

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Doxorubicin Activates ATM-dependent Phosphorylation of Multiple Downstream Targets in Part through the Generation of Reactive Oxygen Species

Ebba U. Kurz, Pauline Douglas, Susan P. Lees‐Miller · Journal of Biological Chemistry · 2004 · 253 citations · Full text

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Promise and challenges in drug discovery and development of hybrid anticancer drugs

Lalji K. Gediya, Vincent C.O. Njar · Expert Opinion on Drug Discovery · 2009 · 220 citations

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