Concepedia

Discovery of novel Tetrahydrobenzo[ b ]thiophene and pyrrole based scaffolds as potent and selective CB2 receptor ligands: The structural elements controlling binding affinity, selectivity and functionality

Noha A. Osman, Alessia Ligresti, Christian D. Klein, Marco Allarà, Alessandro Rabbito, Vincenzo Di Marzo, Khaled A. M. Abouzid

European Journal of Medicinal Chemistry · 2016 · 31 citations · 26 references

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References

26

Molecular characterization of a peripheral receptor for cannabinoids

Sean Munro, Kerrie L. Thomas, Muna Abu-Shaar · Nature · 1993 · 5K citations

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Structure of a cannabinoid receptor and functional expression of the cloned cDNA

Lisa A. Matsuda, Stephen J. Lolait, Michael Brownstein et al. · Nature · 1990 · 5K citations

, , +11

Determination and characterization of a cannabinoid receptor in rat brain.

William A. Devane, F A Dysarz, M R Johnson et al. · Molecular Pharmacology · 1988 · 2.4K citations

Isolation, Structure, and Partial Synthesis of an Active Constituent of Hashish

Yehiel Gaoni, Raphael Mechoulam · Journal of the American Chemical Society · 1964 · 2.4K citations

, , +14

SR 144528, the First Potent and Selective Antagonist of the CB2 Cannabinoid Receptor

M Rinaldi-Carmona, Francis Barth, J Millan et al. · Journal of Pharmacology and Experimental Therapeutics · 1998 · 704 citations · Full text