Dearomatization of Indole Derivatives <i>via</i> Palladium‐Catalyzed CH Bond Functionalization of Pyrroles: Convenient Construction of Spiroindolenines

Abstract

Abstract An intramolecular palladium(II)‐catalyzed dearomative arylation reaction of indoles via CH bond functionalization was developed, providing access to structurally novel spiroindolenines with moderate to good yields. A one‐pot process for the synthesis of spiroindoline derivatives was also realized. magnified image