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Design, synthesis and biological evaluation of 5-amino-4-(1H-benzoimidazol-2-yl)-phenyl-1,2-dihydro-pyrrol-3-ones as inhibitors of protein kinase FGFR1

Andrii Gryshchenko, S. S. Tarnavskiy, Kostiantyn Vasyliovych Levchenko, Volodymyr G. Bdzhola, Galyna P. Volynets, Andriy G. Golub, K.V. Vygranenko, S. M. Yarmoluk

Bioorganic & Medicinal Chemistry · 2016 · 18 citations · 30 references

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30

Rapid colorimetric assay for cellular growth and survival: Application to proliferation and cytotoxicity assays

Tim R. Mosmann · Journal of Immunological Methods · 1983 · 55.6K citations

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AutoDock4 and AutoDockTools4: Automated docking with selective receptor flexibility

Garrett M. Morris, Ruth Huey, William Lindstrom et al. · Journal of Computational Chemistry · 2009 · 25K citations · Full text

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VEGA – An open platform to develop chemo-bio-informatics applications, using plug-in architecture and script programming

Alessandro Pedretti, Luigi Villa, Giulio Vistoli · Journal of Computer-Aided Molecular Design · 2004 · 714 citations

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Targeting FGFR with Dovitinib (TKI258): Preclinical and Clinical Data in Breast Cancer

Fabrice André, Thomas Bachelot, Mario Campone et al. · Clinical Cancer Research · 2013 · 313 citations

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Nuclear translocation of FGFR1 and FGF2 in pancreatic stellate cells facilitates pancreatic cancer cell invasion

Stacey J. Coleman, Athina‐Myrto Chioni, Mohammed Ghallab et al. · EMBO Molecular Medicine · 2014 · 177 citations · Full text

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