Synthesis and antiproliferative evaluation of novel 1,2,4-triazole derivatives incorporating benzisoselenazolone scaffold

Novel thiazolo[3,2-b]-1,2,4-triazoles derived from naproxen with analgesic/anti-inflammatory properties: Synthesis, biological evaluation and molecular modeling studies

Deniz Sarıgöl, Ayşe Uzgören-Baran, Banu Cahide Tel et al. · Bioorganic & Medicinal Chemistry · 2015 · 129 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +15

A randomized phase II study of PX-12, an inhibitor of thioredoxin in patients with advanced cancer of the pancreas following progression after a gemcitabine-containing combination

Ramesh K. Ramanathan, James L. Abbruzzese, Tomislav Dragovich et al. · Cancer Chemotherapy and Pharmacology · 2010 · 119 citations

Medicine, Oncology, Pharmacology +12

Synthesis of novel 1,2,4-triazoles, triazolothiadiazines and triazolothiadiazoles as potential anticancer agents

Mona Kamel, Nadia Y. Megally Abdo · European Journal of Medicinal Chemistry · 2014 · 106 citations

Pharmacy, Medicinal Chemistry, Pharmacology +7

Synthesis and evaluation of benzosuberone embedded with 1,3,4-oxadiazole, 1,3,4-thiadiazole and 1,2,4-triazole moieties as new potential anti proliferative agents

Bandi Yadagiri, S. R. Gurrala, Rajashaker Bantu et al. · Bioorganic & Medicinal Chemistry Letters · 2015 · 93 citations

Pharmacy, Medicinal Chemistry, Pharmacology +12

Synthesis and antitumor activity of 1,2,4-triazoles having 1,4-benzodioxan fragment as a novel class of potent methionine aminopeptidase type II inhibitors

Ya-Ping Hou, Juan Sun, Zhong‐Hua Pang et al. · Bioorganic & Medicinal Chemistry · 2011 · 91 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +7