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Nortropinyl-Arylsulfonylureas as novel, reversible inhibitors of human steroid sulfatase

Peter Nußbaumer, Dieter Geyl, Amarylla Horvath, Philipp Lehr, Barbara Wolff, Andreas Billich

Bioorganic & Medicinal Chemistry Letters · 2003 · 21 citations · 12 references

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12

Estrone sulfamates: potent inhibitors of estrone sulfatase with therapeutic potential

Nicola M. Howarth, Atul Purohit, Michael Reed et al. · Journal of Medicinal Chemistry · 1994 · 218 citations · Full text

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Inactivation of Steroid Sulfatase by an Active Site-Directed Inhibitor, Estrone-3-O-Sulfamate

Atul Purohit, Gary J. Williams, Nicola M. Howarth et al. · Biochemistry · 1995 · 170 citations

, , +13

Sulfamates of various estrogens are prodrugs with increased systemic and reduced hepatic estrogenicity at oral application

W. Elger, Sigfrid Schwarz, Annemarie Hedden et al. · The Journal of Steroid Biochemistry and Molecular Biology · 1995 · 156 citations

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Potent active site-directed inhibition of steroid sulphatase by tricyclic coumarin-based sulphamates

LW Lawrence Woo, Atul Purohit, Bindu Malini et al. · Chemistry & Biology · 2000 · 155 citations · Full text

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2-Substituted 4-(Thio)chromenone 6-<i>O</i>-Sulfamates:  Potent Inhibitors of Human Steroid Sulfatase

Peter Nußbaumer, Philipp Lehr, Andreas Billich · Journal of Medicinal Chemistry · 2002 · 112 citations · Full text

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