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Antitumor Benzothiazoles. 16. Synthesis and Pharmaceutical Properties of Antitumor 2-(4-Aminophenyl)benzothiazole Amino Acid Prodrugs

Ian Hutchinson, S. A. Jennings, B. Rao Vishnuvajjala et al. · Journal of Medicinal Chemistry · 2001 · 420 citations

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Structure-activity relationships of a series of 2-amino-4-thiazole-containing renin inhibitors

William C. Patt, Harriet W. Hamilton, Michael D. Taylor et al. · Journal of Medicinal Chemistry · 1992 · 373 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +15

N-(4-Substituted-thiazolyl)oxamic acid derivatives, new series of potent, orally active antiallergy agents

Karl D. Hargrave, Friedrich K. Hess, James T. Oliver · Journal of Medicinal Chemistry · 1983 · 321 citations

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Synthesis and anti-pseudomonal activity of new 2-isocephems with a dihydroxypyridone moiety at C-7

Koichi Tsuji, Hiroshi Ishikawa · Bioorganic & Medicinal Chemistry Letters · 1994 · 297 citations

Pharmacy, Medicinal Chemistry, Pharmacology +8