Concepedia

Tetrahydroisoquinoline based sulfonamide hydroxamates as potent matrix metalloproteinase inhibitors

Dawei Ma, Wengen Wu, Guoxin Yang, Jingya Li, Jia Li, Qizhuang Ye

Bioorganic & Medicinal Chemistry Letters · 2003 · 34 citations · 22 references

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Discovery of CGS 27023A, a Non-Peptidic, Potent, and Orally Active Stromelysin Inhibitor That Blocks Cartilage Degradation in Rabbits

Lawrence MacPherson, Erol K. Bayburt, Michael Capparelli et al. · Journal of Medicinal Chemistry · 1997 · 325 citations · Full text

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Highly Selective and Orally Active Inhibitors of Type IV Collagenase (MMP-9 and MMP-2):  <i>N</i>-Sulfonylamino Acid Derivatives

Yoshinori Tamura, Fumihiko Watanabe, Takuji Nakatani et al. · Journal of Medicinal Chemistry · 1998 · 283 citations · Full text

, , +10

Inhibition of human skin fibroblast collagenase, thermolysin, and Pseudomonas aeruginosa elastase by peptide hydroxamic acids

Damian Grobelny, Louis Poncz, Richard E. Galardy · Biochemistry · 1992 · 272 citations

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Structure-Based Design of a Novel, Potent, and Selective Inhibitor for MMP-13 Utilizing NMR Spectroscopy and Computer-Aided Molecular Design

James Chen, Frances C. Nelson, Jeremy I. Levin et al. · Journal of the American Chemical Society · 2000 · 107 citations

, , +17

Characterization of a truncated recombinant form of human membrane type 3 matrix metalloproteinase

Taketoshi Shimada, Hiroyuki Nakamura, Eiko Ohuchi et al. · European Journal of Biochemistry · 1999 · 103 citations · Full text

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