Benzo[b]thiophene-2-carboxamides and benzo[b]furan-2-carboxamides are potent antagonists of the human H3-receptor

Auto-inhibition of brain histamine release mediated by a novel class (H3) of histamine receptor

Jean‐Michel Arrang, M. Garbarg, Jean‐Charles Schwartz · Nature · 1983 · 1.6K citations

Life Sciences, Neuroscience, Pharmacology +14

Cloning and Functional Expression of the Human Histamine H₃Receptor

Timothy W. Lovenberg, Barbara Roland, Sandy J. Wilson et al. · Molecular Pharmacology · 1999 · 700 citations · Full text

Life Sciences, Neuroscience, Pharmacology +16

A New Class of Diamine-Based Human Histamine H₃ Receptor Antagonists:  4-(Aminoalkoxy)benzylamines

Richard L. Apodaca, Curt A. Dvorak, Wei Xiao et al. · Journal of Medicinal Chemistry · 2003 · 119 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +14

Diamine-Protonic Acid Catalysts for Catalytic Asymmetric Aldol Reaction

Susumu Saito, Masakazu Nakadai, Hisashi Yamamoto · Synlett · 2001 · 114 citations

Natural Sciences, Chemical Engineering, Chemistry +15

Non-imidazole heterocyclic histamine H3 receptor antagonists

Wenying Chai, J. Guy Breitenbucher, Annette K. Kwok et al. · Bioorganic & Medicinal Chemistry Letters · 2003 · 107 citations · Full text

Medicine, Medicinal Chemistry, Pharmacology +7