Concepedia

Characterization of the Calcitonin Gene-Related Peptide Receptor Antagonist Telcagepant (MK-0974) in Human Isolated Coronary Arteries

Kayi Y. Chan, Lars Edvinsson, Sajedeh Eftekhari, Per Ola Kimblad, Stefanie A. Kane, Joseph J. Lynch, Richard Hargreaves, R. de Vries, Ingrid M. Garrelds, Antoon J. van den Bogaerdt,

Journal of Pharmacology and Experimental Therapeutics · 2010 · 76 citations · 34 references

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References

34

SOME QUANTITATIVE USES OF DRUG ANTAGONISTS

O. ARUNLAKSHANA, H. O. Schild · British Journal of Pharmacology and Chemotherapy · 1959 · 4K citations · Full text

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Contractile properties of small arterial resistance vessels in spontaneously hypertensive and normotensive rats.

Michael J. Mulvany, W Halpern · Circulation Research · 1977 · 2.1K citations

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Calcitonin Gene–Related Peptide Receptor Antagonist BIBN 4096 BS for the Acute Treatment of Migraine

Jes Olesen, Hans‐Christoph Diener, Ingo W. Husstedt et al. · New England Journal of Medicine · 2004 · 1.2K citations · Full text

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The trigeminovascular system and migraine: Studies characterizing cerebrovascular and neuropeptide changes seen in humans and cats

Peter J. Goadsby, Lars Edvinsson · Annals of Neurology · 1993 · 1.2K citations

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Efficacy and tolerability of MK-0974 (telcagepant), a new oral antagonist of calcitonin gene-related peptide receptor, compared with zolmitriptan for acute migraine: a randomised, placebo-controlled, parallel-treatment trial

Tony W. Ho, Michel D. Ferrari, David W. Dodick et al. · The Lancet · 2008 · 529 citations

, , +11