XP13512 [(±)-1-([(α-Isobutanoyloxyethoxy)carbonyl] aminomethyl)-1-cyclohexane Acetic Acid], A Novel Gabapentin Prodrug: I. Design, Synthesis, Enzymatic Conversion to Gabapentin, and Transport by Intestinal Solute Transporters

Kenneth C. Cundy, Russell Branch, Tania Chernov-Rogan, Tracy M. Dias, Toño Estrada, Karin M. Höld, Kerry J. Koller, Xiaoli Liu, Adam Mann, Matt Panuwat,

Journal of Pharmacology and Experimental Therapeutics · 2004 · 151 citations · 32 references

Concepts

References

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