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A practical synthesis of (S) 3-tert-Butoxycarbonylamino-2-oxo-2,3,4,5-tetrahydro-1,5-benzodiazepine-1-acetic acid methyl ester as a conformationally restricted dipeptido-Mimetic for caspase-1 (ICE) inhibitors

David Lauffer, Michael D. Mullican

Bioorganic & Medicinal Chemistry Letters · 2002 · 45 citations · 22 references

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22

Structure and mechanism of interleukin-lβ converting enzyme

Keith P. Wilson, Jo-Anne F. Black, John A. Thomson et al. · Nature · 1994 · 843 citations

, , +11

Peptidomimetics—Tailored Enzyme Inhibitors

Joachim Gante · Angewandte Chemie International Edition in English · 1994 · 817 citations

, , +11

Peptidomimetics for Receptor Ligands—Discovery, Development, and Medical Perspectives

Athanassios Giannis, Thomas Kolter · Angewandte Chemie International Edition in English · 1993 · 778 citations

, , +12

Inactivation of Interleukin-1.beta. Converting Enzyme by Peptide (Acyloxy)methyl Ketones

Nancy A. Thornberry, Erin P. Peterson, Justin J. Zhao et al. · Biochemistry · 1994 · 264 citations

, , +7

Substrate and Inhibitor Specificity of Interleukin-1β-converting Enzyme and Related Caspases

Nara Margolin, Scott A. Raybuck, Keith P. Wilson et al. · Journal of Biological Chemistry · 1997 · 246 citations · Full text

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