Concepedia

Efficient bifunctional gallium-68 chelators for positron emission tomography: tris(hydroxypyridinone) ligands

David J. Berry, Yongmin Ma, James R. Ballinger, Richard Tavaré, Alexander Koers, Kavitha Sunassee, Tao Zhou, Saima Nawaz, Gregory Mullen, Robert C. Hider,

Chemical Communications · 2011 · 138 citations · 17 references

DOI

Concepts

Abstract

A new tripodal tris(hydroxypyridinone) bifunctional chelator for gallium allows easy production of (68)Ga-labelled proteins rapidly under mild conditions in high yields at exceptionally high specific activity and low concentration.

References

17

Radiometal-Labelled Macrocyclic Chelator-Derivatised Somatostatin Analogue with Superb Tumour-Targeting Properties and Potential for Receptor-Mediated Internal Radiotherapy

A. Heppeler, Sylvie Froidevaux, Helmut R. Mäcke et al. · Chemistry - A European Journal · 1999 · 334 citations · Full text

, , +17

Evaluation of Positron Emission Tomography Imaging Using [68Ga]-DOTA-D Phe1-Tyr3-Octreotide in Comparison to [111In]-DTPAOC SPECT. First Results in Patients with Neuroendocrine Tumors

Jeanne Kowalski · Molecular Imaging and Biology · 2003 · 305 citations

, , +14

Metal complexes as diagnostic tools

David E. Reichert, Jason S. Lewis, Carolyn J. Anderson · Coordination Chemistry Reviews · 1999 · 258 citations

, , +12

NODAGATOC, a New Chelator-Coupled Somatostatin Analogue Labeled with [<sup>67/68</sup>Ga] and [<sup>111</sup>In] for SPECT, PET, and Targeted Therapeutic Applications of Somatostatin Receptor (hsst2) Expressing Tumors

Klaus‐Peter Eisenwiener, M. Isabel M. Prata, I. Buschmann et al. · Bioconjugate Chemistry · 2002 · 209 citations

, , +17

Convenient Preparation of <sup>68</sup>Ga-Based PET-Radiopharmaceuticals at Room Temperature

Irina Velikyan, Helmut R. Maëcke, Bengt Långström · Bioconjugate Chemistry · 2008 · 182 citations

, , +17