First synthesis of a strained 14-membered biaryl ether lactone by macrolactonization

The Use of Diethyl Azodicarboxylate and Triphenylphosphine in Synthesis and Transformation of Natural Products

Oyo Mitsunobu · Synthesis · 1981 · 4.1K citations

Natural Sciences, Biochemistry, Chemistry +8

A Rapid Esterification by Means of Mixed Anhydride and Its Application to Large-ring Lactonization

Junji Inanaga, Kuniko Hirata, Hiroko SAEKI et al. · Bulletin of the Chemical Society of Japan · 1979 · 2.2K citations

Natural Sciences, Chemistry, Organic Chemistry +2

Efficient and mild lactonization method for the synthesis of macrolides

E. J. Corey, K. C. Nicolaou · Journal of the American Chemical Society · 1974 · 497 citations

Natural Sciences, Chemistry, Analytical Chemistry +5

Proton-transfer steps in Steglich esterification: a very practical new method for macrolactonization

Eugene P. Boden, Gary E. Keck · The Journal of Organic Chemistry · 1985 · 442 citations

Natural Sciences, Chemistry, Analytical Chemistry +5

Synthesis of macrolides

K. C. Nicolaou · Tetrahedron · 1977 · 295 citations