Vitamin D side chain triazole analogs via cycloaddition `click' chemistry

A Stepwise Huisgen Cycloaddition Process: Copper(I)-Catalyzed Regioselective “Ligation” of Azides and Terminal Alkynes

Vsevolod V. Rostovtsev, Luke G. Green, Valery V. Fokin et al. · Angewandte Chemie International Edition · 2002 · 11.5K citations

Natural Sciences, Chemistry, Catalysis +8

Peptidotriazoles on Solid Phase:  [1,2,3]-Triazoles by Regiospecific Copper(I)-Catalyzed 1,3-Dipolar Cycloadditions of Terminal Alkynes to Azides

Christian W. Tornøe, Caspar Christensen, Morten Meldal · The Journal of Organic Chemistry · 2002 · 8.5K citations

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Direct Synthesis of 1,5-Disubstituted-4-magnesio-1,2,3-triazoles, Revisited

Antoni Krasiński, Valery V. Fokin, K. Barry Sharpless · Organic Letters · 2004 · 271 citations

Pharmacy, Chemistry, Medicinal Chemistry +7

Response of Rat Ventral Prostate to a New and Novel 5αa-Reductase Inhibitor

J. R. Brooks, E.M. Baptista, Charles L. Berman et al. · Endocrinology · 1981 · 145 citations

Life Sciences, Endocrinology, Pharmacology +17

Mechanism of Time-Dependent Inhibition of 5.alpha.-Reductases by .DELTA.1-4-Azasteroids: Toward Perfection of Rates of Time-Dependent Inhibition by Using Ligand-Binding Energies

Gaochao Tian, Robert Mook, Marcia L. Moss et al. · Biochemistry · 1995 · 73 citations

Life Sciences, Biochemistry, Pharmacology +17