Concepedia

Advances in direct C–H arylation of 5,5- 6,5- and 6,6-fused-heterocycles containing heteroatoms (N, O, S)

Saı̈d El Kazzouli, Jamal Koubachi, Nabil El Brahmi, Gérald Guillaumet

RSC Advances · 2015 · 92 citations · 151 references

DOI

Concepts

Abstract

This report aims to review the advances made in C–H arylation of 5,6, 6,6 and 5,5 fused-heterocyclic systems.

References

151

Cu(II)-Catalyzed Direct and Site-Selective Arylation of Indoles Under Mild Conditions

Robert J. Phipps, Neil P. Grimster, Matthew J. Gaunt · Journal of the American Chemical Society · 2008 · 793 citations

, , +12

Room Temperature Palladium-Catalyzed 2-Arylation of Indoles

Nicholas R. Deprez, Dipannita Kalyani, Andrew L. Krause et al. · Journal of the American Chemical Society · 2006 · 646 citations

, , +15

Direct Palladium-Catalyzed C-2 and C-3 Arylation of Indoles:  A Mechanistic Rationale for Regioselectivity

Benjamin S. Lane, Meghann A. Brown, Dalibor Sameš · Journal of the American Chemical Society · 2005 · 645 citations

, , +16

A General Method for Copper-Catalyzed Arylation of Arene C−H Bonds

Hien‐Quang Do, R. Kashif M. Khan, Olafs Daugulis · Journal of the American Chemical Society · 2008 · 593 citations · Full text

, , +13

Establishment of Broadly Applicable Reaction Conditions for the Palladium-Catalyzed Direct Arylation of Heteroatom-Containing Aromatic Compounds

Benoît Liégault, David Lapointe, Laurence Caron et al. · The Journal of Organic Chemistry · 2009 · 591 citations

, , +12