Concepedia

Regio‐ and Enantioselective Aminofluorination of Alkenes

Wangqing Kong, Pascal Feige, Teresa de Haro, Cristina Nevado

Angewandte Chemie International Edition · 2013 · 269 citations · 42 references

DOI

Abstract

Enantio- and regioselective: The intramolecular enantioselective aminofluorination of unactivated olefins was achieved by using a chiral iodo(III) difluoride salt. A highly regioselective aminofluorination of styrenes to access 2-fluoro-2-phenylethanamines was also developed.

References

42

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Enantioselective Formation of Stereogenic Carbon–Fluorine Centers by a Simple Catalytic Method

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, , +15

Enantioselective Kita Oxidative Spirolactonization Catalyzed by In Situ Generated Chiral Hypervalent Iodine(III) Species

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