Concepedia

Recognition of Benztropine by the Dopamine Transporter (DAT) Differs from That of the Classical Dopamine Uptake Inhibitors Cocaine, Methylphenidate, and Mazindol as a Function of a DAT Transmembrane 1 Aspartic Acid Residue

Okechukwu Ukairo, Corry D. Bondi, Amy Hauck Newman, Santosh S. Kulkarni, Alan P. Kozikowski, Stephen Pan, Christopher K. Surratt

Journal of Pharmacology and Experimental Therapeutics · 2005 · 47 citations · 37 references

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37

Cocaine Receptors on Dopamine Transporters Are Related to Self-Administration of Cocaine

Mary C. Ritz, R. J. Lamb, Steven R. Goldberg et al. · Science · 1987 · 2.2K citations

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Conserved aspartic acid residues 79 and 113 of the beta-adrenergic receptor have different roles in receptor function.

Catherine D. Strader, Irving S. Sigal, Mari R. Candelore et al. · Journal of Biological Chemistry · 1988 · 540 citations · Full text

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Dopamine transporter site-directed mutations differentially alter substrate transport and cocaine binding.

S. Kitayama, Shoichi Shimada, H. Eric Xu et al. · Proceedings of the National Academy of Sciences · 1992 · 404 citations

, , +17

Functional Interaction between Monoamine Plasma Membrane Transporters and the Synaptic PDZ Domain–Containing Protein PICK1

Gonzalo E. Torres, Wei-Dong Yao, Amy R. Mohn et al. · Neuron · 2001 · 343 citations · Full text

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-mu opiate receptor. Charged transmembrane domain amino acids are critical for agonist recognition and intrinsic activity.

Christopher K. Surratt, P. S. Johnson, Akiyoshi Moriwaki et al. · Journal of Biological Chemistry · 1994 · 241 citations · Full text

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