Site‐Specific Protein Modification through Cu^<scp>I</scp>‐Catalyzed 1,2,3‐Triazole Formation and Its Implementation in Protein Microarray Fabrication

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Peptidotriazoles on Solid Phase:  [1,2,3]-Triazoles by Regiospecific Copper(I)-Catalyzed 1,3-Dipolar Cycloadditions of Terminal Alkynes to Azides

Christian W. Tornøe, Caspar Christensen, Morten Meldal · The Journal of Organic Chemistry · 2002 · 8.5K citations

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Bioconjugation by Copper(I)-Catalyzed Azide-Alkyne [3 + 2] Cycloaddition

Qian Wang, Timothy R. Chan, Robert Hilgraf et al. · Journal of the American Chemical Society · 2003 · 1.6K citations

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Polytriazoles as Copper(I)-Stabilizing Ligands in Catalysis

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Natural Sciences, Chemistry, Catalysis +10

Cu^I‐Catalyzed Alkyne–Azide “Click” Cycloadditions from a Mechanistic and Synthetic Perspective

Victoria D. Bock, Henk Hiemstra, Jan H. van Maarseveen · European Journal of Organic Chemistry · 2005 · 1.4K citations

Natural Sciences, Chemistry, Catalysis +13