Concepedia

Identification of orally-bioavailable antagonists of the TRPV4 ion-channel

Zhi‐Liang Wei, Margaret Nguyen, Donogh J. R. O’Mahony, Alejandra Acevedo, Sheila Zipfel, Qingling Zhang, Luna Liu, Michelle Dourado, Candace Chi, Victor Yip,

Bioorganic & Medicinal Chemistry Letters · 2015 · 42 citations · 33 references

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33

The capsaicin receptor: a heat-activated ion channel in the pain pathway

Michael J. Caterina, Mark Schumacher, Makoto Tominaga et al. · Nature · 1997 · 9.1K citations

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Vanilloid Receptor–Related Osmotically Activated Channel (VR-OAC), a Candidate Vertebrate Osmoreceptor

Wolfgang Liedtke, Yong Choe, Marc A. Martı́-Renom et al. · Cell · 2000 · 1.4K citations · Full text

, , +7

Anandamide and arachidonic acid use epoxyeicosatrienoic acids to activate TRPV4 channels

Hiroyuki Watanabe, Joris Vriens, Jean Prenen et al. · Nature · 2003 · 1K citations

, , +13

OTRPC4, a nonselective cation channel that confers sensitivity to extracellular osmolarity

Rainer Strotmann, Christian Harteneck, Karin Nunnenmacher et al. · Nature Cell Biology · 2000 · 1K citations

, , +7

Impaired Pressure Sensation in Mice Lacking TRPV4

Makoto Suzuki, Atsuko Mizuno, Kunihiko Kodaira et al. · Journal of Biological Chemistry · 2003 · 737 citations · Full text

, , +17