Structure-activity relationships of synthetic analogs of (-)-epigallocatechin-3-gallate as proteasome inhibitors.

Aslamuzzaman Kazi, Zhigang Wang, Naveen Kumar, Samuel C. Falsetti, Tak Hang Chan, Q. Ping Dou

PubMed · 2004 · 75 citations · 18 references

Abstract

The A-ring and gallate ester/amide bond are essential for the proteasome-inhibitory function of (-)-EGCG.

References

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