Effect of anti-estrogens on the androgen receptor activity and cell proliferation in prostate cancer cells

Cloning of a novel receptor expressed in rat prostate and ovary.

George G. J. M. Kuiper, Eva Enmark, Markku Pelto‐Huikko et al. · Proceedings of the National Academy of Sciences · 1996 · 4.8K citations

Life Sciences, Endocrinology, Molecular Biology +12

A mutation in the ligand binding domain of the androgen receptor of human INCaP cells affects steroid binding characteristics and response to anti-androgens

Jos Veldscholte, C. Ris-Stalpers, George G. J. M. Kuiper et al. · Biochemical and Biophysical Research Communications · 1990 · 945 citations · Full text

Life Sciences, Endocrinology, Molecular Biology +14

Selection for androgen receptor mutations in prostate cancers treated with androgen antagonist.

Mary‐Ellen Taplin, Glenn J. Bubley, Yoo‐Joung Ko et al. · PubMed · 1999 · 599 citations · Full text

Medicine, Oncology, Pharmacology +17

A role for estrogen receptor β in the regulation of growth of the ventral prostate

Sari Mäkelä, Leif C. Andersson, Saija Salmi et al. · Proceedings of the National Academy of Sciences · 2001 · 439 citations · Full text

Life Sciences, Endocrinology, Urology +16

Novel mutations of androgen receptor: a possible mechanism of bicalutamide withdrawal syndrome.

Takahito Hara, Jun‐ichi Miyazaki, Hideo Araki et al. · PubMed · 2003 · 427 citations

Medicine, Endocrinology, Pharmacology +17