Recognition and Transport Characteristics of Nonpeptidic Compounds by Basolateral Peptide Transporter in Caco-2 Cells

Relationship between the inhibition constant (KI) and the concentration of inhibitor which causes 50 per cent inhibition (I50) of an enzymatic reaction

Yung-Chi Cheng, William H. Prusoff · Biochemical Pharmacology · 1973 · 12.8K citations

Cent Inhibition, Inhibitory Activity, Biochemistry +8

Differential Recognition of β-Lactam Antibiotics by Intestinal and Renal Peptide Transporters, PEPT 1 and PEPT 2

Malliga E. Ganapathy, Matthias Brandsch, Puttur D. Prasad et al. · Journal of Biological Chemistry · 1995 · 274 citations · Full text

Cellular Pharmacology, Peptide Science, Antimicrobial Chemotherapy +21

Delta-aminolevulinic acid transport by intestinal and renal peptide transporters and its physiological and clinical implications.

Frank Döring, Justin D. Walter, Jutta Will et al. · Journal of Clinical Investigation · 1998 · 271 citations · Full text

Protein Secretion, Clinical Implications, Gastrointestinal Pharmacology +22

Oral versus intravenous administration of 5-aminolaevulinic acid for photodynamic therapy

C. S. Loh, J Bedwell, N Krasner et al. · British Journal of Cancer · 1993 · 259 citations · Full text

Photochemistry, Photodynamic Therapy, Photobiology +6

Cloning and characterization of a rat H+/peptide cotransporter mediating absorption of beta-lactam antibiotics in the intestine and kidney.

Hideyuki Saito, Masahiro Okuda, Tetsuya Terada et al. · Journal of Pharmacology and Experimental Therapeutics · 1995 · 241 citations