Concepedia

Highly specific, bisubstrate-competitive Src inhibitors from DNA-templated macrocycles

George P. Georghiou, Ralph E. Kleiner, Michael J. Pulkoski‐Gross, David R. Liu, Markus A. Seeliger

Nature Chemical Biology · 2012 · 63 citations · 36 references

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36

[20] Processing of X-ray diffraction data collected in oscillation mode

Zbyszek Otwinowski, W. Minor · Methods in enzymology on CD-ROM/Methods in enzymology · 1997 · 33.6K citations

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<i>Coot</i>: model-building tools for molecular graphics

Paul Emsley, Kevin Cowtan · Acta Crystallographica Section D Biological Crystallography · 2004 · 31.4K citations · Full text

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<i>PHENIX</i>: building new software for automated crystallographic structure determination

Paul D. Adams, Ralf W. Grosse‐Kunstleve, Li‐Wei Hung et al. · Acta Crystallographica Section D Biological Crystallography · 2002 · 4.4K citations · Full text

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A quantitative analysis of kinase inhibitor selectivity

Mazen W. Karaman, Sanna Herrgård, Daniel K. Treiber et al. · Nature Biotechnology · 2008 · 2.4K citations

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Skepinone-L, a Novel Potent and Highly Selective Inhibitor of p38 MAP Kinase, Effectively Impairs Platelet Activation and Thrombus Formation

Oliver Borst, Britta Walker, Patrick Münzer et al. · Cellular Physiology and Biochemistry · 2013 · 1.9K citations · Full text

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