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A-85380 [3-(2(S)-azetidinylmethoxy) pyridine]: In Vitro pharmacological properties of a novel, high affinity α4β2 nicotinic acetylcholine receptor ligand

James P. Sullivan, Diana L. Donnelly‐Roberts, Clark A. Briggs, David J. Anderson, Murali Gopalakrishnan, Marietta Piattoni-Kaplan, Jeffrey E. Campbell, David G. McKenna, Edwardo Molinari, Ann-Marie Hettinger,

Neuropharmacology · 1996 · 137 citations · 34 references

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References

34

Relationship between the inhibition constant (KI) and the concentration of inhibitor which causes 50 per cent inhibition (I50) of an enzymatic reaction

Yung-Chi Cheng, William H. Prusoff · Biochemical Pharmacology · 1973 · 12.9K citations

, , +14

Psychopharmacology: The Fourth Generation of Progress

James J. Brophy · JAMA · 1995 · 1.6K citations

, , +8

Molecular cloning, functional properties, and distribution of rat brain alpha 7: a nicotinic cation channel highly permeable to calcium

Philippe Séguéla, Jacques I. Wadiche, Kelly Dineley‐Miller et al. · Journal of Neuroscience · 1993 · 1.5K citations · Full text

, , +17

Nicotinic binding in rat brain: autoradiographic comparison of [3H]acetylcholine, [3H]nicotine, and [125I]-alpha-bungarotoxin

RD Schwartz, SM Paul, Pert Cb et al. · Journal of Neuroscience · 1985 · 1K citations · Full text

, , +17

α9: An acetylcholine receptor with novel pharmacological properties expressed in rat cochlear hair cells

Ana B. Elgoyhen, David S. Johnson, Jim Boulter et al. · Cell · 1994 · 889 citations

, , +16