Organic Letters · 2006 · 31 citations · 26 references
PharmacyBiochemistryChemistryBiocatalysisDrug DiscoverySynthetic Medicinal ChemistryAmino Acid ChemistryCatalytic MechanismsEnantioselective Synthesis
[reaction: see text] N,N-Dialkyl-beta-amino alcohols derived from alpha-amino acids can be rearranged enantiospecifically by using TFAA/Et3N/NaOH to give 1,2-amino alcohols with enantiomeric excess up to 99%.
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The Synthesis of Vicinal Amino Alcohols
Stephen C. Bergmeier · Tetrahedron · 2000 · 912 citations
Probing the Proteolytic Stability of β‐Peptides Containing α‐Fluoro‐ and α‐Hydroxy‐β‐Amino Acids
David Höök, F. Gessier, Christian Noti et al. · ChemBioChem · 2004 · 131 citations · Full text