Concepedia

Synthesis, pharmacology and molecular modeling of N-substituted 2-phenyl-indoles and benzimidazoles as potent GABAA agonists

José Luis Falcó, Maria Piqué, Miguel A. González, Irma Buira, Eva Méndez, J. Terencio, Cristina Pérez, Marta Príncep, Albert Palomer, Antonio Guglietta

European Journal of Medicinal Chemistry · 2006 · 72 citations · 7 references

DOI

Concepts

References

7

Experimental and computational approaches to estimate solubility and permeability in drug discovery and development settings

Christopher A. Lipinski, Franco Lombardo, Beryl W. Dominy et al. · Advanced Drug Delivery Reviews · 1997 · 11.2K citations

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Comprehensive Medicinal Chemistry

Quantitative Structure-Activity Relationships · 1991 · 749 citations

2-Aryl-3-indoleacetamides (FGIN-1): a new class of potent and specific ligands for the mitochondrial DBI receptor (MDR).

Elena Romeo, James Auta, Alan P. Kozikowski et al. · Journal of Pharmacology and Experimental Therapeutics · 1992 · 156 citations · Full text

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Participation of mitochondrial diazepam binding inhibitor receptors in the anticonflict, antineophobic and anticonvulsant action of 2-aryl-3-indoleacetamide and imidazopyridine derivatives.

James Auta, Elena Romeo, Alan P. Kozikowski et al. · Journal of Pharmacology and Experimental Therapeutics · 1993 · 57 citations

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Tolerance to Anticonvulsant Effects of Diazepam, Clonazepam, and Clobazam in Amygdala‐Kindled Rats

Howard C. Rosenberg, Elizabeth I. Tietz, Ted H. Chiu · Epilepsia · 1989 · 48 citations

, , +11