Concepedia

DPI-3290 [(+)-3-((α-R)-α-((2 S,5 R)-4-Allyl-2,5-dimethyl-1-piperazinyl)-3-hydroxybenzyl)-N-(3-fluorophenyl)-N-methylbenzamide]. II. A Mixed Opioid Agonist with Potent Antinociceptive Activity and Limited Effects on Respiratory Function

Peter J. Gengo, Hugh O. Pettit, Scott J. O’Neill, Ying Su, Robert W. McNutt, Kwen‐Jen Chang

Journal of Pharmacology and Experimental Therapeutics · 2003 · 26 citations · 19 references

DOI

Concepts

References

19

The Pharmacological Basis of Therapeutics

American Journal of Health-System Pharmacy · 1976 · 8.2K citations

, , +10

Opioid analgesics and antagonists

Terry Reisine · Medical Entomology and Zoology · 1996 · 1.2K citations

, , +12

Classification of multiple morphine and enkephalin binding sites in the central nervous system.

Benjamin Wolozin, Gavril W. Pasternak · Proceedings of the National Academy of Sciences · 1981 · 372 citations

, , +16

Differential stereochemical requirements of mu vs. delta opioid receptors for ligand binding and signal transduction: development of a class of potent and highly delta-selective peptide antagonists.

Peter W. Schiller, Tin Nguyen, Grazyna Weltrowska et al. · Proceedings of the National Academy of Sciences · 1992 · 240 citations · Full text

, , +17

A novel, potent and selective nonpeptidic delta opioid receptor agonist BW373U86.

K J Chang, Greg C. Rigdon, J. L. Howard et al. · Journal of Pharmacology and Experimental Therapeutics · 1993 · 162 citations

, , +17