European Journal of Medicinal Chemistry · 2014 · 16 citations · 11 references
PharmacyMedicinal ChemistryPharmacologyDrug DiscoveryMolecular PharmacologyStructure-activity RelationshipsEnzyme InhibitionLead Compound DesignPotency OptimizationStructure-activity Relationship AnalysisTyrosine Kinase InhibitorsBiological Evaluation ReportKinase InhibitorsPyrimidine AnalogsPyrimidine AnaloguesPyrimidine ChemistryRos1 InhibitorsRos1-targeted Therapy
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Identifying and Targeting <i>ROS1</i> Gene Fusions in Non–Small Cell Lung Cancer
Kurtis D. Davies, Anh T. Le, Mariana F. Theodoro et al. · Clinical Cancer Research · 2012 · 472 citations · Full text
Acquired Resistance to Crizotinib from a Mutation in <i>CD74</i>–<i>ROS1</i>
Mark M. Awad, Ryohei Katayama, Michele McTigue et al. · New England Journal of Medicine · 2013 · 413 citations · Full text
Medicine, Oncology, Pharmacology +17
Edward G. Shaw, Meihua Wang, Stephen W. Coons et al. · Journal of Clinical Oncology · 2012 · 354 citations
Óscar de Frutos, Carmen Atienza, Antonio M. Echavarren · European Journal of Organic Chemistry · 2001 · 43 citations