Functional Characterization of an Organic Cation Transporter (hOCT1) in a Transiently Transfected Human Cell Line (HeLa)

Relationship between the inhibition constant (KI) and the concentration of inhibitor which causes 50 per cent inhibition (I50) of an enzymatic reaction

Yung-Chi Cheng, William H. Prusoff · Biochemical Pharmacology · 1973 · 12.9K citations

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Drug excretion mediated by a new prototype of polyspecific transporter

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Cloning and Characterization of Two Human Polyspecific Organic Cation Transporters

Valentin Gorboulev, Jochen C. Ulzheimer, Aida Akhoundova et al. · DNA and Cell Biology · 1997 · 636 citations · Full text

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Cloning and characterization of a novel human pH‐dependent organic cation transporter, OCTN1

Ikumi Tamai, Hikaru Yabuuchi, Jun-ichi Nezu et al. · FEBS Letters · 1997 · 458 citations

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Cloning and Functional Expression of a Human Liver Organic Cation Transporter

Lei Zhang, Mark J. Dresser, Andrew T. Gray et al. · Molecular Pharmacology · 1997 · 417 citations · Full text

Life Sciences, Biochemistry, Molecular Biology +10