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FLUORINATED 2-(4-AMINO-3-METHYLPHENYL)BENZOTHIAZOLES INDUCE CYP1A1 EXPRESSION, BECOME METABOLIZED, AND BIND TO MACROMOLECULES IN SENSITIVE HUMAN CANCER CELLS

Eileen Brantley, Valentina Trapani, Michael C. Alley, Curtis Hose, Tracey D. Bradshaw, Malcolm F. G. Stevens, Edward A. Sausville, Sherman F. Stinson

Drug Metabolism and Disposition · 2004 · 53 citations · 32 references

DOI

Concepts

References

32

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The anti-malarial artesunate is also active against cancer

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Antitumor Benzothiazoles. 14. Synthesis and in Vitro Biological Properties of Fluorinated 2-(4-Aminophenyl)benzothiazoles

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