Diversity‐Oriented Three‐Component Reactions of Diazo Compounds with Anilines and 4‐Oxo‐Enoates

Changcheng Jing, Dong Xing, Yu Qian, Taoda Shi, Yun Zhao, Wenhao Hu

Angewandte Chemie International Edition · 2013 · 74 citations · 25 references

Concepts

Abstract

Choosing a path: The title reaction can proceed through two different reaction pathways, and is controlled by the addition sequence of the substrates. Divergent polyfunctional products, pyrrolidines or linear α-amino ester derivatives, are obtained in good yields and high diastereoselectivities.

References

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