Design, synthesis, and biological evaluation of novel 2-pyridinyl-[1,2,4]triazoles as inhibitors of transforming growth factor β1 type 1 receptor

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Direct binding of Smad3 and Smad4 to critical TGFβ‐inducible elements in the promoter of human plasminogen activator inhibitor‐type 1 gene

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TGFβ signals through a heteromeric protein kinase receptor complex

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Structural basis of inhibitor selectivity in MAP kinases

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