Discovery of a 2,4-Disubstituted Pyrrolo[1,2-<i>f</i>][1,2,4]triazine Inhibitor (BMS-754807) of Insulin-like Growth Factor Receptor (IGF-1R) Kinase in Clinical Development - Concepedia

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Discovery of a 2,4-Disubstituted Pyrrolo[1,2-<i>f</i>][1,2,4]triazine Inhibitor (BMS-754807) of Insulin-like Growth Factor Receptor (IGF-1R) Kinase in Clinical Development

DOI Full Paper Access

94

Citations

8

References

2009

Year

Mark D. Wittman, Joan M. Carboni, Yang Zheng, Francis Y. Lee, Melissa Antman, Ricardo M. Attar, Praveen Balimane, ChiehYing Chang, Cliff Chen, Lorell Discenza,

Journal of Medicinal Chemistry

Abstract

This report describes the biological activity, characterization, and SAR leading to 9d (BMS-754807) a small molecule IGF-1R kinase inhibitor in clinical development.

References

	Year	Citations

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