TRPV4 activation triggers the release of melatonin from human non-pigmented ciliary epithelial cells

N-((1 S)-1-{[4-((2 S)-2-{[(2,4-Dichlorophenyl)sulfonyl]amino}-3-hydroxypropanoyl)-1-piperazinyl]carbonyl}-3-methylbutyl)-1-benzothiophene-2-carboxamide (GSK1016790A), a Novel and Potent Transient Receptor Potential Vanilloid 4 Channel Agonist Induces Urinary Bladder Contraction and Hyperactivity: Part I

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Medicine, Pharmacology, Physiology +16

Identification and characterization of novel TRPV4 modulators

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Pharmacy, Medicinal Chemistry, Molecular Biology +4

Melatonin uptake through glucose transporters: a new target for melatonin inhibition of cancer

David Hevia, Pedro González‐Menéndez, Isabel Quirós-González et al. · Journal of Pineal Research · 2015 · 144 citations · Full text

Medicine, Oncology, Pharmacology +12

Involvement of melatonin MT3 receptors in the regulation of intraocular pressure in rabbits

Jesús Pintor, Laura Martin, Teresa Peláez et al. · European Journal of Pharmacology · 2001 · 123 citations

Medicine, Ophthalmology, Physiology +13

The Ciliary Body - The Third Organ Found to Synthesize Indoleamines in Humans

Xavier D. Martin, Halina Z Malina, Mary C. Brennan et al. · European Journal of Ophthalmology · 1992 · 112 citations

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