Structure–activity relationships for dipeptide prodrugs of acyclovir: Implications for prodrug design

9-(2-Hydroxyethoxymethyl)guanine activity against viruses of the herpes group

H. J. Schaeffer, Lilia M. Beauchamp, P de Miranda et al. · Nature · 1978 · 1.1K citations

Medicine, Virology, Herpes Group +3

Comparative Efficacy of Antiherpes Drugs against Different Strains of Herpes Simplex Virus

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Transport of Valganciclovir, a Ganciclovir Prodrug, via Peptide Transporters PEPT1 and PEPT2

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Synthesis and antiviral activity of water-soluble esters of acyclovir [9-[(2-hydroxyethoxy)methyl]guanine)

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Cellular Uptake Mechanism of Amino Acid Ester Prodrugs in Caco-2/hPEPT1 Cells Overexpressing a Human Peptide Transporter

Hyo-Kyung Han, Doo‐Man Oh, Gordon L. Amidon · Pharmaceutical Research · 1998 · 95 citations · Full text