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Synthesis and structure–activity relationships of piperidinylpyrrolopyridine derivatives as potent and selective H1 antagonists

Sı́lvia Fonquerna, M. Miralpeix, Lluı́s Pagès, Carles Puig, Arantxa Cardús, Francisca Antón, Dolors Vilella, Mònica Aparici, Graham J. Warrellow, Jörge Beleta,

Bioorganic & Medicinal Chemistry Letters · 2005 · 16 citations · 5 references

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5

Binding characteristics of 3H-prazosin to rat brain α-adrenergic receptors

Pamela Greengrass, Rona Bremmer · European Journal of Pharmacology · 1979 · 419 citations · Full text

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HETEROGENEITY OF HISTAMINE Hi‐RECEPTORS: SPECIES VARIATIONS IN [<sup>3</sup>H]MEPYRAMINE BINDING OF BRAIN MEMBRANES

Raymond S.L. Chang, Vinh T. Tran, Solomon H. Snyder · Journal of Neurochemistry · 1979 · 223 citations

, , +14

Mesulergine, a selective serotonin-2 ligand in the rat cortex, does not label these receptors in porcine and human cortex: Evidence for species differences in brain serotonin-2 receptors

Ángel Pazos, Daniël Hoyer, José Palacios · European Journal of Pharmacology · 1984 · 138 citations

, , +17

Synthesis and Structure−Activity Relationships of Novel Histamine H<sub>1</sub> Antagonists:  Indolylpiperidinyl Benzoic Acid Derivatives

Sı́lvia Fonquerna, M. Miralpeix, Lluı́s Pagès et al. · Journal of Medicinal Chemistry · 2004 · 23 citations · Full text

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Comparative study of central and peripheral histamine‐H<sub>1</sub> receptor binding in vitro and ex vivo of non‐sedating antihistamines and of noberastine, a new agent

Josée E. Leysen, W Gommeren, Paul F.M. Janssen et al. · Drug Development Research · 1991 · 16 citations

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