Concepedia

Studies of the Biogenic Amine Transporters. XI. Identification of a 1-[2-[Bis(4-fluorophenyl)methoxy]ethyl]-4-(3-phenylpropyl)piperazine (GBR12909) Analog That Allosterically Modulates the Serotonin Transporter

Barbara Nightingale, Christina M. Dersch, Terrence L. Boos, Elisabeth Greiner, William J. Calhoun, Arthur E. Jacobson, Kenner C. Rice, Richard B. Rothman

Journal of Pharmacology and Experimental Therapeutics · 2005 · 18 citations · 21 references

References

21

Amphetamine-type central nervous system stimulants release norepinephrine more potently than they release dopamine and serotonin

Richard B. Rothman, Michael H. Baumann, Christina M. Dersch et al. · Synapse · 2000 · 931 citations · Full text

Medicine, Neuroscience, Pharmacology +17

The kinetics of competitive radioligand binding predicted by the law of mass action.

Harvey Motulsky, L C Mahan · Molecular Pharmacology · 1984 · 419 citations

Medicine, Chemistry, Pharmacology +17

SSRIs and SNRIs: broad spectrum of efficacy beyond major depression.

Justine Kent · PubMed · 1999 · 132 citations

Pharmacy, Pharmacotherapy, Psychiatry +17

Sildenafil for Iatrogenic Serotonergic Antidepressant Medication-Induced Sexual Dysfunction in 4 Patients

H. George Nurnberg, John Lauriello, Paula L. Hensley et al. · The Journal of Clinical Psychiatry · 1999 · 129 citations

Medicine, Pharmacology, Pharmacotherapy +16

Labeling by [3H]1,3-di(2-tolyl)guanidine of two high affinity binding sites in guinea pig brain: evidence for allosteric regulation by calcium channel antagonists and pseudoallosteric modulation by sigma ligands.

RB Rothman, Audrey A. Reid, Artin Mahboubi et al. · Molecular Pharmacology · 1991 · 112 citations

Medicine, Neurobiology, Pharmacology +10