Stereoselective total synthesis of topographically constrained designer amino acids: 2′, 6′-dimethyl-β-methyltyrosines

Conformation and Biological Activity of Cyclic Peptides

Horst Kessler · Angewandte Chemie International Edition in English · 1982 · 868 citations

Natural Sciences, Biochemistry, Biophysics +16

The asymmetric synthesis of .alpha.-amino acids. Electrophilic azidation of chiral imide enolates, a practical approach to the synthesis of (R)- and (S)-.alpha.-azido carboxylic acids

David A. Evans, Thomas C. Britton, Jonathan A. Ellman et al. · Journal of the American Chemical Society · 1990 · 451 citations

Natural Sciences, Chemistry, Organic Chemistry +13

Conformational restrictions of biologically active peptides via amino acid side chain groups

Victor J. Hruby · Life Sciences · 1982 · 399 citations

Life Sciences, Biochemistry, Molecular Biology +16

Asymmetric glycine enolate aldol reactions: synthesis of cyclosporin's unusual amino acid, MeBmt

David A. Evans, Ann E. Weber · Journal of the American Chemical Society · 1986 · 343 citations

Natural Sciences, Biochemistry, Medicinal Chemistry +8

The asymmetric synthesis of β-lactam antibiotics - I. application of chiral oxazolidones in the staudinger reaction.

David A. Evans, Eric B. Sjogren · Tetrahedron Letters · 1985 · 205 citations

Pharmacy, Medicinal Chemistry, Drug Discovery +8