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MedicinePharmacokineticsPharmacologyNeuropharmacologyBlood-brain Barrier PenetrationBlood-brain Barrier PharmacologySerotonergic PharmacologyAntihistamine PharmacologyCerebral Drug PenetrationEx Vivo ModelsHistamine Receptor AntagonismHistamine Receptor AntagonistsHistamine Receptor PharmacologyHistamine Receptors
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Highly potent and selective ligands for histamine H3-receptors
J.M. Arrang, M. Garbarg, J.-C. Lancelo et al. · Nature · 1987 · 902 citations
Jane Clapham, Gavin J. Kilpatrick · British Journal of Pharmacology · 1992 · 260 citations · Full text
Medicine, Neuroscience, Pharmacology +17