Synthesis, characterization and anti-microbial studies of some novel 2,4-disubstituted thiazoles

Phenethylthiazolethiourea (PETT) Compounds, a New Class of HIV-1 Reverse Transcriptase Inhibitors. 1. Synthesis and Basic Structure-Activity Relationship Studies of PETT Analogs

Frank W. Bell, Amanda Cantrell, Marita Hoegberg et al. · Journal of Medicinal Chemistry · 1995 · 455 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +15

Structure-activity relationships of a series of 2-amino-4-thiazole-containing renin inhibitors

William C. Patt, Harriet W. Hamilton, Michael D. Taylor et al. · Journal of Medicinal Chemistry · 1992 · 373 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +15

N-(4-Substituted-thiazolyl)oxamic acid derivatives, new series of potent, orally active antiallergy agents

Karl D. Hargrave, Friedrich K. Hess, James T. Oliver · Journal of Medicinal Chemistry · 1983 · 321 citations

Pharmacy, Medicinal Chemistry, Pharmacology +9

Synthesis and anti-pseudomonal activity of new 2-isocephems with a dihydroxypyridone moiety at C-7

Koichi Tsuji, Hiroshi Ishikawa · Bioorganic & Medicinal Chemistry Letters · 1994 · 297 citations

Pharmacy, Medicinal Chemistry, Pharmacology +8

4-(1,2,5,6-Tetrahydro-1-alkyl-3-pyridinyl)-2-thiazolamines: a novel class of compounds with central dopamine agonist properties

Juan C. Jaén, Lawrence D. Wise, Bradley W. Caprathe et al. · Journal of Medicinal Chemistry · 1990 · 255 citations · Full text

Medicine, Medicinal Chemistry, Pharmacology +17