Efficient coupling of α,α-dimethyl amino acid using a new chloro imidazolidium reagent, CIP

1-Hydroxy-7-azabenzotriazole. An efficient peptide coupling additive

Louis A. Carpino · Journal of the American Chemical Society · 1993 · 1.5K citations

Natural Sciences, Chemistry, Pharmacology +7

PyBOP® and PyBroP: Two reagents for the difficult coupling of the α,α-dialkyl amino acid, Aib.

Eric Frérot, J. H. Coste, Antoine Pantaloni et al. · Tetrahedron · 1991 · 227 citations

Pharmacy, Biochemistry, Medicinal Chemistry +3

Comparative study of methods to couple hindered peptides

Jeffrey R. Spencer, Valery V. Antonenko, Nancy G. J. Delaet et al. · International journal of peptide & protein research · 1992 · 75 citations

Natural Sciences, Biochemistry, Medicinal Chemistry +14

Self-indicating activated esters for use in solid phase peptide synthesis. Fluorenylmethoxycarbonylamino acid derivatives of 3-hydroxy-4-oxodihydrobenzotriazine

Eric Atherton, Linda R. Cameron, Morten Meldal et al. · Journal of the Chemical Society Chemical Communications · 1986 · 53 citations

Natural Sciences, Chemistry, Organic Chemistry +7

Emerimicins III and IV and their ethylalanine12 epimers. Facilitated chemical-enzymatic synthesis and a qualitative evaluation of their solution structures

Urszula Słomczyńska, Denise D. Beusen, Janusz Zabrocki et al. · Journal of the American Chemical Society · 1992 · 47 citations

Natural Sciences, Biochemistry, Chemistry +6